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Neurotransmitter Transporter Inhibitors Library

10,813 compounds

Neurotransmitter Transporter Inhibitors Library is a set of small-molecule inhibitors. They are used to treat mental disorders.

Protein Tyrosine Phosphatase Non-receptor Type (PTPN) Targeted Library

32,596 compounds

PTPN Targeted Library is a set of small-molecule inhibitors. Protein tyrosine phosphatases are important signaling molecules in cell proliferation.

GPCR Targeted Library

29,185 compounds

Small-molecule compounds that can be used in GPCR drug discovery. Dysregulation of these receptors causes diabetes, CNS disorders.

Protein Kinases Inhibitors Library

36,324 compounds

Protein Kinases Inhibitors Library is modulators that are used in cancer and inflammation treatment.

DGK Inhibitors Library

10,674 compounds

Diacylglycerol kinase Inhibitors Library is a set of small-molecules that can inhibit the progression of cancer and innate cytotoxic immunocytes.

Ligand-Gated Ion Channels Library

3,743 compounds

Ligand-Gated Ion Channels Library is a set of small-molecule compounds that target LGICs. They can be used in the treatment of neurodegenerative disorders.

Carbonic Anhydrase II Library

5,000 compounds

Carbonic anhydrase II library is a set of compounds belonging to the sulfonamides, mercaptans and phenols aimed at modulating of Carbonic anhydrase II activity

NOTUM (Wnt signaling) Library

4,003 compounds

Small molecules that can inhibit NOTUM thus potentially treating diseases caused by dysregulation of Wnt signaling.

RAR (Nuclear receptors) Ligands Library

6,767 compounds

Set of RAR receptor antagonists. The retinoic acid receptor is a type of nuclear receptor which can also act as a transcription factor.

Proline Kinase Library

2,081 compounds

Proline Kinase Library is a set of kinase inhibitors. These kinases play a crucial role in diverse cellular processes and human diseases.

15,080 compounds

Molecules from c-Met Library target receptor tyrosine kinase. It prevents binding hepatocyte growth factor with c-Met which can lead to cancer.

Serine Proteases Inhibitors Library

31,972 compounds

Serine Proteases Inhibitors Library is a set of small-molecule compounds that target serine proteases and can be used in anticancer drug discovery.

Protein Arginine Methyltransferases Library

27,102 compounds

PRMT Library is set of small-molecule compounds with reported affinity against cancer-assosiated PRMTs.

Receptor protein tyrosine phosphatases

3,765 compounds

RPTP Targeted Library is small-molecule inhibitors. Disruption of protein tyrosine phosphorylation contributes to a variety of human diseases.

Ion Channels Focused Library

26,421 compounds

Ion Channels Focused Library is small-molecule compounds selected for modulating ion channels proteins. They are therapeutic targets of CNS diseases.

Cysteine Proteases Inhibitors Library

7,801 compounds

Set of small-molecule compounds that can target cysteine proteases and be used in drug development for cancer, viral, infections treatment.

Androgen Receptor Antagonists Library

4,244 compounds

Androgen Receptor Antagonists Library is a set of non-steroidal small molecules for prostate cancer treatment.

KRAS-Targeted Library

16,000 compounds

KRAS-Targeted Library is a set of novel KRAS-active compounds.

Arginase Targeted Library

2,016 compounds

Arginase Targeted Library is a set of small-molecule compounds against arginase. This enzyme is implicated in cancer immunosuppression and tumor growth.

Aurora A-B Kinases Targeted Library

9,342 compounds

Set of small-molecule serine/threonine kinases family inhibitors.

PI3K-Targeted Library

16,720 compounds

PI3K-Targeted Library is a set of small-molecule inhibitors of PI3K signaling pathway. They can be used in effective inhibiting tumor progression.

PD-1/L1 Library

PD-1/L1 Library is a set of PD-1 and PD-L1 inhibitors. It is a group of anticancer drugs that block the activity of immune checkpoint proteins.

Glucocorticoid receptors Library

4,768 compounds

Glucocorticoid Receptors Library is small-molecule selective modulators of GR which regulates gene transcription.

Adenosine Receptors Targeted Library

19,626 compounds

Adenosine Receptors Targeted Library is a set of small-molecule ligands. They can be used for treating neurodegeneration diseases.

7,123 compounds

Set of GABA receptor antagonists. These drug-like compounds inhibit the action of GABA and produce stimulant and convulsant effects.

Purinergic Library

3,271 compounds

Purinergic Library is a set of purinergic receptor antagonists. Such antagonists are used for thrombosis and stroke treatment.

TLR-8 ligands Library

TLR-8 Ligands Library is a set of small-molecule TLR-8 agonists. They can be used in adjuvantation research and for the treatment of ovarian cancer.

Type II Kinase Inhibitors Library

6,996 compounds

Type II Kinase Inhibitors Library is a set of non-ATP site inhibitors or activators that bind to an extended ATP site including a back pocket.

Developmental Pathway (Hh/Wnt) Set

2,230 compounds

Developmental Pathway Hh/Wnt Set is inhibitors of the Hedgehog and Wnt-signaling pathways implicated in cancer.

Allosteric Kinases Inhibitors Library

22,697 compounds

Small‐molecule allosteric kinase modulators that target allosteric pockets of kinases outside the conserved ATP‐binding pocket.

BRD4 Targeted Library

4,462 compounds

BRD4 Targeted Library is a set of small-molecule compounds that inhibit transcriptional and epigenetic regulator - BRD4.

Indoleamine 2,3-dioxygenase 1 Focused Library

5,601 compounds

Indoleamine 2,3-dioxygenase1 Focused Library is a set of small-molecule compounds that can inhibit inappropriate IDO activity in tumours.

Integrin Receptors Targeted library

1,708 compounds

Integrin Receptors Targeted library is a set of RGD peptides or peptidomimetics that affect many events in tumor cells thereby directly induce apoptosis.

Neuropeptide S Library

2,800 compounds

Neuropeptide S Library is a set of small-molecule NPSR ligands. They can be used in psychiatric disorders treatment as anxiolytics and analgesics.

Chelators targeting matrix metalloproteinases library

8,600 compounds

Chelators targeting matrix metalloproteinases are small-molecule that inhibit proteolytic activity of tumor cells and prevent metastasis.

Voltage-Gated Ion Channel-Targeted Library

4,723 compounds

Voltage-Gated Ion Channel-Targeted set is small molecule compounds that contribute to treating pain.

STING Agonist Library

5,939 compounds

STING Agonist Library is small-molecules that bind and activate STING and lead to IFN production. Can be used in cancer immunotherapy.

Chemokine Receptor-Targeted Library

18,150 compounds

Chemokine Receptor Targeted Library is a set of small-molecule ligands. Modulation of chemokine receptor is used in the treatment of inflammatory diseases.

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