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Protein Tyrosine Phosphatase Non-receptor Type (PTPN) Targeted Library

33,000 compounds

PTPN Targeted Library is a set of small-molecule inhibitors. Protein tyrosine phosphatases are important signaling molecules in cell proliferation.

Protein Kinases Inhibitors Library

38,000 compounds

Protein Kinases Inhibitors Library is modulators that are used in cancer and inflammation treatment.

PD-1/L1 Library

PD-1/L1 Library is a set of PD-1 and PD-L1 inhibitors. It is a group of anticancer drugs that block the activity of immune checkpoint proteins.

Ion Channels Focused Library

26,000 compounds

Ion Channels Focused Library is small-molecule compounds selected for modulating ion channels proteins. They are therapeutic targets of CNS diseases.

Arginase Targeted Library

2,000 compounds

Arginase Targeted Library is a set of small-molecule compounds against arginase. This enzyme is implicated in cancer immunosuppression and tumor growth.

Receptor protein tyrosine phosphatases

3,900 compounds

RPTP Targeted Library is small-molecule inhibitors. Disruption of protein tyrosine phosphorylation contributes to a variety of human diseases.

RAR (Nuclear receptors) Ligands Library

6,000 compounds

Nuclear receptors Ligands Library is a set of RAR receptor antagonists. The retinoic acid receptor is a type of nuclear receptor which can also act as a transcription factor.

Cysteine Proteases Inhibitors Library

8,000 compounds

Cysteine Proteases Inhibitors Library is a set of small-molecule compounds that can be used in drug development for cancer, viral, infections treatment.

GPCR Targeted Library

40,000 compounds

G protein-coupled receptors Targeted Library is small-molecule compounds that can be used in GPCR drug discovery. Dysregulation of these receptors causes diabetes, CNS disorders.

Chelators targeting matrix metalloproteinases library

9,300 compounds

Chelators targeting matrix metalloproteinases are small-molecule that inhibit proteolytic activity of tumor cells and prevent metastasis.

Neurotransmitter Transporter Inhibitors library

12,000 compounds

Neurotransmitter Transporter Inhibitors Library is a set of reuptake inhibitors. They are used to treat mental disorders.

Serine Proteases Inhibitors Library

37,000 compounds

Serine Proteases Inhibitors Library is a set of small-molecule compounds that target serine proteases and can be used in anticancer drug discovery.

Protein Arginine Methyltransferases Library

31,000 compounds

PRMT Library is set of small-molecule compounds with reported affinity against cancer-assosiated PRMTs.

Purinergic Library

3,500 compounds

Purinergic Library is a set of purinergic receptor antagonists. Purinergic signaling is mediated by ATP. Such antagonists is used for thrombosis treatment.

Androgen Receptor Antagonists Library

4,300 compounds

Androgen Receptor Antagonists Library is a set of non-steroidal small-molecules for prostate cancer treatment.

Proline Kinase Library

2,000 compounds

Proline Kinase Library is a set of kinase inhibitors. These kinases play a crucial role in diverse cellular processes and human diseases.

Adenosine Receptors Targeted Library

21,000 compounds

Adenosine Receptors Targeted Library is a set of small-molecule ligands. They can be used for treating neurodegeneration diseases.

PI3K-Targeted Library

19,000 compounds

PI3K-Targeted Library is a set of small-molecule inhibitors of PI3K signaling pathway. They can be used in effective inhibiting tumor progression.

Allosteric Kinases Inhibitors Library

26,000 compounds

Small‐molecule allosteric kinase inhibitors bind to an allosteric site outside the conserved ATP‐binding pocket overcoming poor selectivity of kinase inhibitors.

Type II Kinase Inhibitors Library

8,000 compounds

Type II Kinase Inhibitors Library is a set of non-ATP site inhibitors or activators that bind to an extended ATP site including a back pocket.

Ligand-Gated Ion Channels Library

4,000 compounds

Ligand-Gated Ion Channels Library is a set of small-molecule compounds that target LGICs. They can be used in the treatment of neurodegenerative disorders.

Integrin Receptors Targeted library

2,000 compounds

Integrin Receptors Targeted library is a set of RGD peptides or peptidomimetics that affect many events in tumor cells thereby directly induce apoptosis.

STING Agonist Library

6,000 compounds

STING Agonist Library is small-molecules that bind and activate STING and lead to IFN production. Can be used in cancer immunotherapy.

16,000 compounds

Molecules from c-Met Library target receptor tyrosine kinase. It prevents binding hepatocyte growth factor with c-Met which can lead to cancer.

KRAS-Targeted Library

11,000 compounds

KRAS-Targeted Library is a set of novel KRAS-active compounds. The small G-proteins KRas function as GDP–GTP regulated binary switches in many signal transduction pathways.

Developmental Pathway (Hh/Wnt) Set

2,000 compounds

Developmental Pathway Hh/Wnt Set is inhibitors of the Hedgehog and Wnt-signaling pathways implicated in cancer.

7,271 compounds

gamma-Aminobutyric acid Library is a set of GABAA receptor antagonists. These drug-like compounds inhibit the action of GABA and produce stimulant and convulsant effects.

Aurora A-B Kinases Library

10,000 compounds

Aurora A-B Kinases Library is a set of small-molecule serine/threonine kinases family inhibitors. Overexpression of Aurora kinases is clarified in a number of cancers.

Glucocorticoid receptors Library

5,000 compounds

Glucocorticoid Receptors Library is small-molecule selective modulators of GR which regulates gene transcription.

DGK Inhibitors Library

12,000 compounds

Diacylglycerol kinase Inhibitors Library is a set of small-molecules that can inhibit the progression of cancer and innate cytotoxic immunocytes.

Voltage-Gated Ion Channel-Targeted Library

5,000 compounds

Voltage-Gated Ion Channel-Targeted set is small molecule compounds that contribute to treating pain.

TLR-8 ligands Library

TLR-8 Ligands Library is a set of small-molecule TLR-8 agonists. They can be used in adjuvantation research and for the treatment of ovarian cancer.

BRD4 Targeted Library

5,000 compounds

BRD4 Targeted Library is a set of small-molecule compounds that inhibit transcriptional and epigenetic regulator - BRD4.

Indoleamine 2,3-dioxygenase 1 Focused Library

6,000 compounds

Indoleamine 2,3-dioxygenase1 Focused Library is a set of small-molecule compounds that can inhibit inappropriate IDO activity in tumours.

Neuropeptide S Library

3,000 compounds

Neuropeptide S Library is a set of small-molecule NPSR ligands. They can be used in psychiatric disorders treatment as anxiolytics and analgesics.

Chemokine Receptor-Targeted Library

20,000 compounds

Chemokine Receptor Targeted Library is a set of small-molecule ligands. Modulation of chemokine receptor is used in the treatment of inflammatory diseases.

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